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Anton Simeonov
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Journal Articles

Fatty Acid Derivatization and Cyclization of the Immunomodulatory Peptide RP-182 Targeting CD206high Macrophages Improve Antitumor Activity

Open Access
Sitanshu S. Singh, Raul Calvo, Anju Kumari, Rushikesh V. Sable, Yuhong Fang, Dingyin Tao, Xin Hu, Sarah Gray Castle, Saifun Nahar, Dandan Li, Emily Major, Tino W. Sanchez, Rintaro Kato, Xin Xu, Jian Zhou, Liang Liu, Christopher A. LeClair, Anton Simeonov, Bolormaa Baljinnyam, Mark J. Henderson, Juan Marugan, Udo Rudloff
Journal: Molecular Cancer Therapeutics
Mol Cancer Ther (2024) 23 (12): 1827–1841.
https://doi.org/10.1158/1535-7163.MCT-23-0790
Published: 03 December 2024
View articletitled, Fatty Acid Derivatization and Cyclization of the Immunomodulatory Peptide RP-182 Targeting CD206high Macrophages Improve Antitumor Activity
Open the PDF for Fatty Acid Derivatization and Cyclization of the Immunomodulatory Peptide RP-182 Targeting CD206high Macrophages Improve Antitumor Activity in another window
Includes: Supplementary data
Journal Articles

KDM5B Promotes Drug Resistance by Regulating Melanoma-Propagating Cell Subpopulations

Free
Xiaoni Liu, Shang-Min Zhang, Meaghan K. McGeary, Irina Krykbaeva, Ling Lai, Daniel J. Jansen, Stephen C. Kales, Anton Simeonov, Matthew D. Hall, Daniel P. Kelly, Marcus W. Bosenberg, Qin Yan
Journal: Molecular Cancer Therapeutics
Mol Cancer Ther (2019) 18 (3): 706–717.
https://doi.org/10.1158/1535-7163.MCT-18-0395
Published: 01 March 2019
View articletitled, KDM5B Promotes Drug Resistance by Regulating Melanoma-Propagating Cell Subpopulations
Open the PDF for KDM5B Promotes Drug Resistance by Regulating Melanoma-Propagating Cell Subpopulations in another window
Includes: Supplementary data
Journal Articles

Biochemical Assays for the Discovery of TDP1 Inhibitors

Free
Christophe Marchand, Shar-yin N. Huang, Thomas S. Dexheimer, Wendy A. Lea, Bryan T. Mott, Adel Chergui, Alena Naumova, Andrew G. Stephen, Andrew S. Rosenthal, Ganesha Rai, Junko Murai, Rui Gao, David J. Maloney, Ajit Jadhav, William L. Jorgensen, Anton Simeonov, Yves Pommier
Journal: Molecular Cancer Therapeutics
Mol Cancer Ther (2014) 13 (8): 2116–2126.
https://doi.org/10.1158/1535-7163.MCT-13-0952
Published: 05 August 2014
View articletitled, Biochemical Assays for the Discovery of TDP1 Inhibitors
Open the PDF for Biochemical Assays for the Discovery of TDP1 Inhibitors in another window
Includes: Supplementary data
Journal Articles

Abstract A168: Quantitative high‐throughput screening for inhibitors of human apurinic/apyrimidinic endonuclease APE1

Free
Dorjbal Dorjsuren, Ajit Jadhav, Avanti Kulkarni, Daniel McNeill, Christopher P. Austin, David M. Wilson, III, Min Shen, Anton Simeonov
Journal: Molecular Cancer Therapeutics
Mol Cancer Ther (2009) 8 (12_Supplement): A168.
https://doi.org/10.1158/1535-7163.TARG-09-A168
Published: 10 December 2009
View articletitled, Abstract A168: Quantitative high‐throughput screening for inhibitors of human apurinic/apyrimidinic endonuclease APE1
Journal Articles

Identification of phosphotyrosine mimetic inhibitors of human tyrosyl-DNA phosphodiesterase I by a novel AlphaScreen high-throughput assay

Free
Christophe Marchand, Wendy A. Lea, Ajit Jadhav, Thomas S. Dexheimer, Christopher P. Austin, James Inglese, Yves Pommier, Anton Simeonov
Journal: Molecular Cancer Therapeutics
Mol Cancer Ther (2009) 8 (1): 240–248.
https://doi.org/10.1158/1535-7163.MCT-08-0878
Published: 12 January 2009
View articletitled, Identification of phosphotyrosine mimetic inhibitors of human tyrosyl-DNA phosphodiesterase I by a novel AlphaScreen high-throughput assay
Open the PDF for Identification of phosphotyrosine mimetic inhibitors of human tyrosyl-DNA phosphodiesterase I by a novel AlphaScreen high-throughput assay in another window
Includes: Supplementary data